Phenylmorphans

[borohydride]

http://oasys2.confex.com/acs/236nm/techprogram/images/1184906-0.gif

The above is a widely studied class of opioids. Example 2 is around x 500 morphine in potency. The question is - would they be considered analogues under the CsA act? Of course, one would expect the N-(2-furanylethyl) analogue to be still stronger...

[thesimple]

this is interesting, would love to know more about whether they are covered.

[borohydride]

They appear to be legal but they are a bit of a pain to make. I think they are interesting because if you overlay them with ketobemidone - they do so very well - I guess that is why the =O & =CH2 are the strong ones.

If you want legal then almost any phenolic opioid can have the -OH replaced with a -CONH2 and keep the same activity (and duration goes up a huge amount - the M analogue lasts 14 hours or more).

I'm not getting more into the simpler but unusual opioids. AH-7921 was a washout but there are some sneaky nortilidine analogues that seem about x10M (and are legal).

[Frenchy0707]

Sure wish I had any fucking idea what you are talking about Boro. ^^^^It's all Greek to me. I flunked chemistry:(